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Obituary
Yoshito Kishi (1937-2023)
Yoshito Kishi (1937-2023)
Professor. Yoshito Kishi,
a member of the Honorary Editorial Associates of HETEROCYCLES,
has passed away on January 9, 2023 at the age of 85.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
January 13, 2023
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Paper | Special issue | Vol 95, No. 2, 2017, pp.787-798
Published online, 1st November, 2016
Published online, 1st November, 2016
DOI: 10.3987/COM-16-S(S)42
■ Triphosgene-Mediated Chlorolactamization and Aminolactamization of Homoallylic Amines
Yuika Nishida, Norihiko Takeda, Okiko Miyata,* and Masafumi Ueda*
*Department of Medicinal Chemistry, Kobe Pharmaceutical University, 4-19-1, Motoyamakitamachi, Higashinada, Kobe 658-8558, Japan
Abstract
Two types of aminocarbonylation reaction of homoallylic amines have been developed. The treatment of homoallylic amines with triphosgene in dichloromethane led to formation of the corresponding β-chlorolactams via Prins-type cyclization of a carbamoyl chloride intermediate. For the reaction in acetonitrile, β-aminolactams were obtained via sequential Prins-type cyclization and Ritter-type reactions.
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