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Obituary
Zenichi Yoshida (1925-2023)
Zenichi Yoshida (1925-2023)
Professor. Zenichi Yoshida,
a member of the Honorary Advisors of HETEROCYCLES (1975-1998),
has passed away on May 4, 2023 at the age of 97.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
May 11, 2023
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Review | Regular issue | Vol 91, No. 8, 2015, pp.1555-1577
Published online, 14th July, 2015
Published online, 14th July, 2015
DOI: 10.3987/REV-15-822
■ Synthesis and Bioactivity of Pyrroloindazoles: An Overview
Manas Chakrabarty,* Moumita Rakshit, and Gandhi K Kar
*Department of Chemistry, Presidency University, 86/1, College Street, Kolkata-700073, India
Abstract
In this review, the synthesis and bioactivity of pyrroloindazoles have been presented. The pyrroloindazoles were synthesised either by the heteroannulation of tetrahydro-indolones/isoindolones, aminoindazoles, Sonogashira/Cacchi indazolic substrates or acyl/aroylindole ketoxime dinitrophenyl ethers or by the cycloaddition of indolynes, indazolic betaines, styrylpyrazoles and nitroindazoles. Several pyrroloindazoles showed analgesic, antiinflammatory and antitumor properties, inhibition of Pim kinase and soluble guanylate cyclase, and antagonism of NMDA-receptor.
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