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Obituary
Zenichi Yoshida (1925-2023)
Zenichi Yoshida (1925-2023)
Professor. Zenichi Yoshida,
a member of the Honorary Advisors of HETEROCYCLES (1975-1998),
has passed away on May 4, 2023 at the age of 97.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
May 11, 2023
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Review | Regular issue | Vol 92, No. 9, 2016, pp.1561-1597
Published online, 5th August, 2016
Published online, 5th August, 2016
DOI: 10.3987/REV-16-844
■ Efficient Synthesis of Heterocycles Using Highly Electrophilic Ethenetricarboxylates
Shoko Yamazaki*
*Department of Chemistry, Nara University of Education, Takabatake-cho, Nara 630-8528, Japan
Abstract
The synthesis of heterocyclic compounds utilizing highly electrophilic ethenetricarboxylates is described. Ethenetricarboxylate is a member of methylenemalonates and more reactive than frequently used alkylidenemalonates by the electron-withdrawing effect of 2-carboxyl group. They are utilized as efficient Michael acceptors or electron-deficient C=C components. Lewis acids also promote the reactions of ethenetricarboxylate derivatives efficiently. The intermolecular and intramolecular reactions of ethenetricarboxylates towards synthesis of heterocycles are presented.
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