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Obituary
Yoshito Kishi (1937-2023)
Yoshito Kishi (1937-2023)
Professor. Yoshito Kishi,
a member of the Honorary Editorial Associates of HETEROCYCLES,
has passed away on January 9, 2023 at the age of 85.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
January 13, 2023
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Paper | Regular issue | Vol 83, No. 3, 2011, pp.555-570
Published online, 26th January, 2011
Published online, 26th January, 2011
DOI: 10.3987/COM-10-12115
■ Friedel-Crafts Reactions of Vinylaziridine Linked to an Ester Group
Hisashi Takada, Eiko Yasui, Yui Sahara, Yūki Chinen, Hirotoshi Tanaka, Yusuke Morita, Chihiro Kobiki, Daiki Narisawa, Megumi Mizukami, Masaaki Miyashita, and Shinji Nagumo*
*Department of Applied Chemistry, Faculty of Engineering, Kogakuin University, Nakano 2665-1, Hachioji, Tokyo, 192-0015, Japan
Abstract
Intermolecular Friedel-Crafts reactions of vinylaziridines 11, 12, 15, 16 and 20 linked to an ester with various benzene derivatives occurred at the C4 position selectively to afford 5-amino-4-aryl-2-hexenoate derivatives in good yields.
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