HETEROCYCLES
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Obituary
Zenichi Yoshida (1925-2023)
Zenichi Yoshida (1925-2023)
Professor. Zenichi Yoshida,
a member of the Honorary Advisors of HETEROCYCLES (1975-1998),
has passed away on May 4, 2023 at the age of 97.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
May 11, 2023
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1980
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Paper | Regular issue | Vol 78, No. 1, 2009, pp.59-70
Published online, 25th August, 2008■ Synthesis of Azole Derivatives from 3-Phenylaminopropanhydrazide and Evaluation of Their Antimicrobial Efficacy
Published online, 25th August, 2008
DOI: 10.3987/COM-08-11478
■ Synthesis of Azole Derivatives from 3-Phenylaminopropanhydrazide and Evaluation of Their Antimicrobial Efficacy
Ingrida Tumosiene, Kristina Kantminiene, Alvydas Pavilonis, Zaneta Mazeliene, and Zigmuntas J. Beresnevicius*
*Department of Organic Chemistry, Kaunas University of Technology, Radvilenu pl. 19, Kaunas LT-50254, Lithuania
Abstract
Novel pyrrole and pyrazole derivatives containing phenylaminopropanoyl moiety were synthesized from 3-phenylaminopropanohydrazide through its condensation with diketones. The intramolecular cyclization reaction of disubstituted semicarbazides and thiosemicarbazides was used to prepare new 1,3,4-thiadiazole, 1,3,4-oxadiazole and 1,2,4-triazole compounds. Some of the synthesized compounds were evaluated for in vitro antimicrobial activity.
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