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Note | Regular issue | Vol 48, No. 9, 1998, pp.1935-1941
Published online, 1st January, 1970
DOI: 10.3987/COM-98-8261
Reactions of 2-tert-Butyl-3-phenyl-oxaziridine with Alkyl Isothiocyanates and Its Application to Glucosyl-aminoheterocycle Synthesis

Masao Shimizu,* Yasuo Gama, and Isao Shibuya

*National Institute of Advanced Industrial Science and Technology, 1-1-1 Higashi, Tsukuba, Ibaraki 305-8565, Japan


2-tert-Butyl-3-phenyloxaziridine was heated with alkyl isothiocyanates to afford 4-alkyl-2-tert-butyl-3-phenyl-1,2,4-oxadiazolidine-5-thiones. The reaction mechanism of the ring formation was discussed. This reaction was applicable to synthesis of glucosylaminoheterocycles.