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Obituary
Yoshito Kishi (1937-2023)
Yoshito Kishi (1937-2023)
Professor. Yoshito Kishi,
a member of the Honorary Editorial Associates of HETEROCYCLES,
has passed away on January 9, 2023 at the age of 85.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
January 13, 2023
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Paper | Regular issue | Vol 41, No. 10, 1995, pp.2279-2287
Published online, 1st January, 1970■ A New Synthesis of 3-Substituted Indolines and Indoles
Published online, 1st January, 1970
DOI: 10.3987/COM-95-7177
■ A New Synthesis of 3-Substituted Indolines and Indoles
Masaru Kihara,* Yasumasa Iwai, and Yoshimitsu Nagao
*Faculty of Pharmaceutical Sciences, University of Tokushima, Sho-machi, Tokushima 770, Japan
Abstract
3-Phenyl- and 3-alkyl-3-hydroxyindolines were synthesized by intramolecular Barbier reaction of phenyl and alkyl N-(2-iodophenyl)-N-methylaminomethyl ketones with n-BuLi, which were easily prepared from N-methyl-2-iodoaniline and bromomethyl ketones. The treatment of the indolines with acid gave the corresponding indoles in quantitative yields.
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