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Paper | Special issue | Vol 35, No. 1, 1993, pp.193-204
Published online, 1st January, 1970
DOI: 10.3987/COM-92-S6
Synthesis and Reactions of 4-(α-Aminoarylidene)thiazetidine 1,1-Dioxides

Herbert Plagge and Hans-Hartwig Otto*

*Pharmazeutisches Institut, LS Pharmazeutische Chemie, Albert-Ludwigs-Universität Freiburg, Hermann-Herder-Str. 9 D-7800 Freiburg i.Br., Germany


β-Sultams react as highly potent sulfonyl analogues of β-lactams with aromatic nitriles to the title compounds (2). Hydrolysis, reduction, and reactions of 2 with acylating and alkylating agents are described. Some of the compounds show a week β-lactamase inhibition.