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Yoshito Kishi (1937-2023)
Yoshito Kishi (1937-2023)
Professor. Yoshito Kishi,
a member of the Honorary Editorial Associates of HETEROCYCLES,
has passed away on January 9, 2023 at the age of 85.
I deeply express my regret over his death.
Kunio Ogasawara
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January 13, 2023
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Paper | Regular issue | Vol 36, No. 4, 1993, pp.733-742
Published online, 1st January, 1970■ A Convenient Synthesis of 5-Substituted Tetrahydro-1,4,3-oxathiazine 4,4-Dioxides
Published online, 1st January, 1970
DOI: 10.3987/COM-92-6207
■ A Convenient Synthesis of 5-Substituted Tetrahydro-1,4,3-oxathiazine 4,4-Dioxides
Evelyne Grunder-Klotz,* Paul Humbert, and Jean-Daniel Ehrhardt
*Laboratoire de Pharmacologie Cardiovasculaire et Rénale, URA 589 CNRS, Université Louis Pasteur, 11 rue Humann, F-67000 Strasbourg, France
Abstract
An advantageous one pot procedure for the synthesis of tetrahydro-1,4,3-oxathiazine 4,4-dioxides by dialkylation of readily available α,N-alkyl- or arylsulfonamide dianions with gaseous formaldehyde is reported. Stability and some reactions of these heterocycles are also described.
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