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Obituary
Yoshito Kishi (1937-2023)
Yoshito Kishi (1937-2023)
Professor. Yoshito Kishi,
a member of the Honorary Editorial Associates of HETEROCYCLES,
has passed away on January 9, 2023 at the age of 85.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
January 13, 2023
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Paper | Regular issue | Vol 53, No. 12, 2000, pp.2739-2751
Published online, 1st January, 1970■ Stereoselective Synthesis of 4(5)-[(2S,3S)- and (2R,3R)-3-Aminotetrahydrofuran-2-yl)imidazoles Using Modified and Standard Mitsunobu Cyclizations: Synthetic Studies toward Novel Histamine H3-Ligands
Published online, 1st January, 1970
DOI: 10.3987/COM-00-9052
■ Stereoselective Synthesis of 4(5)-[(2S,3S)- and (2R,3R)-3-Aminotetrahydrofuran-2-yl)imidazoles Using Modified and Standard Mitsunobu Cyclizations: Synthetic Studies toward Novel Histamine H3-Ligands
Shinya Harusawa, Ikuno Ijichi, Lisa Araki, and Takushi Kurihara*
*Osaka University of Pharmaceutical Sciences, 4-20-1 Nasahara, Takatsuki, Osaka 569-1094, Japan
Abstract
4(5)-[(2S,3S)-3-Aminotetrahydrofuran-2-yl)imidazole [(+)-3] and its enantiomer [(-)-(2R,3R)-3] were stereoselectivity synthesized by using both modified and standard Mitsunobu cyclizations from L- and D-methionine, respectively.
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