

HETEROCYCLES
An International Journal for Reviews and Communications in Heterocyclic ChemistryWeb Edition ISSN: 1881-0942
Published online by The Japan Institute of Heterocyclic Chemistry
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Natural Products with Heterocyclic Ring System
Structure
New Heterocyclic Natural Products
Updated: 26 June, 2015
This journal will list the new natural products with a heterocyclic ring system, collected from current chemical literature, whose structure has been established.
- Search by Group: AllPolyketidesAromaticsTerpenesSteroidsAlkaloidsAntibioticsMiscellaneous
- Search by Journal: Chem. Pharm. Bull.Helv. Chim. ActaHeterocyclesJ. Antibiot.J. Nat. Prod.J. Org. Chem.Org. Biomol. Chem.Org. Lett.Phytochem. Lett.PhytochemistryPlanta medicaTetrahedronTetrahedron Lett.
- Year: 2014201420142014201420142014201420142014201420142014
- Vol: 6297896777791216107107807055
- No: 11111111112143, 4421, 22 1744-4745-48
Terpenes
Asperulogenin
C10H12O4 = 196
Helv. Chim. Acta 2014, 97, 1571
H. Kırmızıbekmez, H. Bardakcı,
M. Masullo, Ö. Kamburoğlu,
G. Eryılmaz, G. Akaydın,
E. Yeşilada, S. Piacente
DOI: 10.1002/hlca.201400065
CrossRef
[ | NS | ] | Asperula lilaciflora | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 10.4 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Russulanobiline A
C15H20O3 = 248
Phytochemistry 2014, 107, 126
O. Malagòn, A. Porta, M. Clericuzio,
G. Gilardoni, D. Gozzini, G. Vidari
DOI: 10.1016/j.phytochem.2014.08.018
CrossRef
[ | NS | ] | Russula nobilis | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 181.2 [ CH2Cl2 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Russulanobiline B
C15H20O3 = 248
Phytochemistry 2014, 107, 126
O. Malagòn, A. Porta, M. Clericuzio,
G. Gilardoni, D. Gozzini, G. Vidari
DOI: 10.1016/j.phytochem.2014.08.018
CrossRef
[ | NS | ] | Russula nobilis | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 295.5 [ CH2Cl2 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Russulanobiline C
C15H18O4 = 262
Phytochemistry 2014, 107, 126
O. Malagòn, A. Porta, M. Clericuzio,
G. Gilardoni, D. Gozzini, G. Vidari
DOI: 10.1016/j.phytochem.2014.08.018
CrossRef
[ | NS | ] | Russula nobilis | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 154.5 [ CH2Cl2 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
No Name
C20H30O4 = 334
J. Nat. Prod. 2014, 77, 2342
Z.-Y. Wu, Y.-B. Zhang, K.-K. Zhu,
C. Luo, J.-X. Zhang, C.-R. Cheng,
R.-H. Feng, W.-Z. Yang, F. Zeng,
Y. Wang, P.-P. Xu, J.-L. Guo, X. Liu,
S.-H. Guan, D.-A. Guo
DOI: 10.1021/np500125x
CrossRef
[ | NS | ] | Acanthopanax gracilistylus | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 24 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] | inhibit effect of IL-8 |
Terpenes
Rhizomucronol A
C20H32O4 = 336
Helv. Chim. Acta 2014, 97, 1531
A. Madhu, A. S. C. V. A. Rao,
S. Sushma, P. M. Gowri,
T. V. Raju
DOI: 10.1002/hlca.201400022
CrossRef
[ | NS | ] | Rhizophora mucronata | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | – 125 [ CHCl3 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Rhizomucronol B
C20H32O4 = 336
Helv. Chim. Acta 2014, 97, 1531
A. Madhu, A. S. C. V. A. Rao,
S. Sushma, P. M. Gowri,
T. V. Raju
DOI: 10.1002/hlca.201400022
CrossRef
[ | NS | ] | Rhizophora mucronata | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | – 105 [ CHCl3 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Heterophyllin C, Hydroperoxy-
C17H22O7 = 338
Chem. Pharm. Bull. 2014, 62, 1092
Y. Saito, T. Mukai, Y. Iwamoto,
M. Baba, K. Takiguchi, Y. Okamoto,
X. Gong, T. Kawahara, C. Kuroda,
M. Tori
DOI: 10.1248/cpb.c14-00426
CrossRef
[ | NS | ] | Eupatorium heterophyllum | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 14.5 [ CHCl3 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Holophyllin A
C20H30O5 = 350
Tetrahedron Lett. 2014, 55, 6504
C. S. Kim, B. Shin, O. W. Kwon,
S. Y. Kim, S. U. Choi, D.-C. Oh,
K. H. Kim, K. R. Lee
DOI: 10.1016/j.tetlet.2014.10.030
CrossRef
[ | NS | ] | Abies holophylla | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | – 12.3 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] | inhibitory activity against NO production |
Terpenes
Heterophyllin A, Keto-
C20H24O7 = 376
Chem. Pharm. Bull. 2014, 62, 1092
Y. Saito, T. Mukai, Y. Iwamoto,
M. Baba, K. Takiguchi, Y. Okamoto,
X. Gong, T. Kawahara, C. Kuroda,
M. Tori
DOI: 10.1248/cpb.c14-00426
CrossRef
[ | NS | ] | Eupatorium heterophyllum | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 109.9 [ CHCl3 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Kuguacin U
C25H36O5 = 416
Helv. Chim. Acta 2014, 97, 1546
J.-C. Chen, X.-X. Yuan, L. Zhou,
J.-Q. Liu, Y. Nian, Z.-R. Li, Y. Li,
M.-J. Xie, M.-H. Qiu
DOI: 10.1002/hlca.201400051
CrossRef
[ | NS | ] | Momordica charantia | ||||||||
[ | mp | ] | 295 - 296 ℃ | ||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 14.8 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Heterophyllin H, Hydroperoxy-
C22H28O8 = 420
Chem. Pharm. Bull. 2014, 62, 1092
Y. Saito, T. Mukai, Y. Iwamoto,
M. Baba, K. Takiguchi, Y. Okamoto,
X. Gong, T. Kawahara, C. Kuroda,
M. Tori
DOI: 10.1248/cpb.c14-00426
CrossRef
[ | NS | ] | Eupatorium heterophyllum | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 33.2 [ CHCl3 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Heterophyllin B, Hydroperoxy-
C22H28O9 = 436
Chem. Pharm. Bull. 2014, 62, 1092
Y. Saito, T. Mukai, Y. Iwamoto,
M. Baba, K. Takiguchi, Y. Okamoto,
X. Gong, T. Kawahara, C. Kuroda,
M. Tori
DOI: 10.1248/cpb.c14-00426
CrossRef
[ | NS | ] | Eupatorium heterophyllum | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 13.8 [ CHCl3 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Phyllaemblicin G3
C22H28O9 = 436
Org. Biomol. Chem. 2014, 12, 8764
J.-J. Lv, Y.-F. Wang, J.-M. Zhang,
S. Yu, D. Wang, H.-T. Zhu,
R.-R. Cheng, C.-R. Yang, M. Xu,
Y.-J. Zhang
DOI: 10.1039/C4OB01196A
CrossRef
[ | NS | ] | Phyllanthus emblica | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 31.3 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Heterophyllin A, Hydroperoxy-
C22H28O10 = 452
Chem. Pharm. Bull. 2014, 62, 1092
Y. Saito, T. Mukai, Y. Iwamoto,
M. Baba, K. Takiguchi, Y. Okamoto,
X. Gong, T. Kawahara, C. Kuroda,
M. Tori
DOI: 10.1248/cpb.c14-00426
CrossRef
[ | NS | ] | Eupatorium heterophyllum | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 19.9 [ CHCl3 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Kuguacin V
C30H46O4 = 470
Helv. Chim. Acta 2014, 97, 1546
J.-C. Chen, X.-X. Yuan, L. Zhou,
J.-Q. Liu, Y. Nian, Z.-R. Li, Y. Li,
M.-J. Xie, M.-H. Qiu
DOI: 10.1002/hlca.201400051
CrossRef
[ | NS | ] | Momordica charantia | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | – 26.6 [ Py. ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Kuguacin W
C30H46O4 = 470
Helv. Chim. Acta 2014, 97, 1546
J.-C. Chen, X.-X. Yuan, L. Zhou,
J.-Q. Liu, Y. Nian, Z.-R. Li, Y. Li,
M.-J. Xie, M.-H. Qiu
DOI: 10.1002/hlca.201400051
CrossRef
[ | NS | ] | Momordica charantia | ||||||||
[ | mp | ] | 113 - 115 ℃ | ||||||||
[ | bp | ] | |||||||||
[ | α | ] D | – 15.7 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Heterophyllin E, Hydroperoxy-
C24H30O10 = 478
Chem. Pharm. Bull. 2014, 62, 1092
Y. Saito, T. Mukai, Y. Iwamoto,
M. Baba, K. Takiguchi, Y. Okamoto,
X. Gong, T. Kawahara, C. Kuroda,
M. Tori
DOI: 10.1248/cpb.c14-00426
CrossRef
[ | NS | ] | Eupatorium heterophyllum | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 62.0 [ EtOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Heterophyllin G, Hydroperoxy-
C24H30O10 = 478
Chem. Pharm. Bull. 2014, 62, 1092
Y. Saito, T. Mukai, Y. Iwamoto,
M. Baba, K. Takiguchi, Y. Okamoto,
X. Gong, T. Kawahara, C. Kuroda,
M. Tori
DOI: 10.1248/cpb.c14-00426
CrossRef
[ | NS | ] | Eupatorium heterophyllum | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 5.6 [ EtOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Hexatenuin B
C31H44O4 = 480
Tetrahedron 2014, 70, 8312
A. Umeyama, C. Ohta, Y. Shino,
M. Okada, Y. Nakamura,
T. Hamagaki, H. Imagawa,
M. Tanaka, A. Ishiyama,
M. Iwatsuki, K. Otoguro, S. Ōmura,
T. Hashimoto
DOI: 10.1016/j.tet.2014.09.013
CrossRef
[ | NS | ] | Hexagonia tenuis | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 189 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] | antitrypanosomal activity |
Terpenes
Kuguacin T
C30H46O5 = 486
Helv. Chim. Acta 2014, 97, 1546
J.-C. Chen, X.-X. Yuan, L. Zhou,
J.-Q. Liu, Y. Nian, Z.-R. Li, Y. Li,
M.-J. Xie, M.-H. Qiu
DOI: 10.1002/hlca.201400051
CrossRef
[ | NS | ] | Momordica charantia | ||||||||
[ | mp | ] | 193 - 195 ℃ | ||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 1.1 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Heterophyllin D, Hydroperoxy-
C24H30O11 = 494
Chem. Pharm. Bull. 2014, 62, 1092
Y. Saito, T. Mukai, Y. Iwamoto,
M. Baba, K. Takiguchi, Y. Okamoto,
X. Gong, T. Kawahara, C. Kuroda,
M. Tori
DOI: 10.1248/cpb.c14-00426
CrossRef
[ | NS | ] | Eupatorium heterophyllum | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 6.9 [ EtOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Heterophyllin F, Hydroperoxy-
C24H30O11 = 494
Chem. Pharm. Bull. 2014, 62, 1092
Y. Saito, T. Mukai, Y. Iwamoto,
M. Baba, K. Takiguchi, Y. Okamoto,
X. Gong, T. Kawahara, C. Kuroda,
M. Tori
DOI: 10.1248/cpb.c14-00426
CrossRef
[ | NS | ] | Eupatorium heterophyllum | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 17.2 [ EtOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Nimbolinin C, 1-Decinnamoyl-
C29H40O8 = 516
Phytochemistry 2014, 107, 175
G.-Y. Zhu, L.-P. Bai, L. Liu,
Z.-H. Jiang
DOI: 10.1016/j.phytochem.2014.08.009
CrossRef
[ | NS | ] | Melia toosendan | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 73.0 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Havanensin 3,12-Diacetate, 14,15-Deoxy-11-oxo-
C30H40O8 = 528
Phytochemistry 2014, 107, 175
G.-Y. Zhu, L.-P. Bai, L. Liu,
Z.-H. Jiang
DOI: 10.1016/j.phytochem.2014.08.009
CrossRef
[ | NS | ] | Melia toosendan | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 28.1 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] | TNFα-induced NF-κB luciferase activity |
Terpenes
Volkensin, 3-Deacetyl-12-O-methyl-
C32H44O8 = 556
Phytochemistry 2014, 107, 175
G.-Y. Zhu, L.-P. Bai, L. Liu,
Z.-H. Jiang
DOI: 10.1016/j.phytochem.2014.08.009
CrossRef
[ | NS | ] | Melia toosendan | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 33.1 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Trichilinin, 11,15-Dioxo-
C30H38O10 = 558
Phytochemistry 2014, 107, 175
G.-Y. Zhu, L.-P. Bai, L. Liu,
Z.-H. Jiang
DOI: 10.1016/j.phytochem.2014.08.009
CrossRef
[ | NS | ] | Melia toosendan | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 12.9 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Swielimonoid A
C32H38O9 = 566
J. Nat. Prod. 2014, 77, 2367
Y.-B. Cheng, Y.-T. Chien, J.-C. Lee,
C.-K. Tseng, H.-C. Wang, I-W. Lo,
Y.-H. Wu, S.-Y. Wang, Y.-C. Wu,
F.-R. Chang
DOI: 10.1021/np5002829
CrossRef
[ | NS | ] | Swietenia macrophylla | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | + 23 [ CH2Cl2 ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |
Terpenes
Hexatenuin A
C34H48O7 = 568
Tetrahedron 2014, 70, 8312
A. Umeyama, C. Ohta, Y. Shino,
M. Okada, Y. Nakamura,
T. Hamagaki, H. Imagawa,
M. Tanaka, A. Ishiyama,
M. Iwatsuki, K. Otoguro, S. Ōmura,
T. Hashimoto
DOI: 10.1016/j.tet.2014.09.013
CrossRef
[ | NS | ] | Hexagonia tenuis | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 208 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] | antitrypanosomal activity |
Terpenes
Nimbolinin C, 1-Decinnamoyl-1-(2’-methylacryloyl)-
C33H44O9 = 584
Phytochemistry 2014, 107, 175
G.-Y. Zhu, L.-P. Bai, L. Liu,
Z.-H. Jiang
DOI: 10.1016/j.phytochem.2014.08.009
CrossRef
[ | NS | ] | Melia toosendan | ||||||||
[ | mp | ] | |||||||||
[ | bp | ] | |||||||||
[ | α | ] D | - 5.8 [ MeOH ] | ||||||||
[ | Ph | ] |
|
||||||||
[ | act | ] |